Melanotan II studies: 324 papers with results
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- Cloning, tissue distribution, pharmacology and three-dimensional modelling of melanocortin receptors 4 and 5 in rainbow trout suggest close evolutionary relationship of these subtypes.
Haitina T · The Biochemical journal · 2004
In vitro (cells) · rainbow trout (receptor) · 1 result
- Biological and conformational examination of stereochemical modifications using the template melanotropin peptide, Ac-Nle-c[Asp-His-Phe-Arg-Trp-Ala-Lys]-NH2, on human melanocortin receptors.
Haskell-Luevano C · Journal of medicinal chemistry · 1997
In vitro (cells) · 1 result
- The melanocortin receptor subtypes in chicken have high preference to ACTH-derived peptides.
Ling MK · British journal of pharmacology · 2004
In vitro (cells) · chicken · 1 result
- Conformation of the core sequence in melanocortin peptides directs selectivity for the melanocortin MC3 and MC4 receptors.
Oosterom J · The Journal of biological chemistry · 1999
In vitro (cells) · 2 results
- Pharmacological characterization of 30 human melanocortin-4 receptor polymorphisms with the endogenous proopiomelanocortin-derived agonists, synthetic agonists, and the endogenous agouti-related protein antagonist.
Xiang Z · Biochemistry · 2010
In vitro (cells) · 1 result
- Characterizations of the unusual dissociation properties of melanotropin peptides from the melanocortin receptor, hMC1R.
Haskell-Luevano C · Journal of medicinal chemistry · 1996
In vitro (cells) · 3 results
- Molecular cloning, characterization and brain mapping of the melanocortin 5 receptor in the goldfish.
Cerdá-Reverter JM · Journal of neurochemistry · 2003
In vitro (cells) · goldfish · 1 result
- ARPE-19-derived VEGF-containing exosomes promote neovascularization in HUVEC: the role of the melanocortin receptor 5.
Maisto R · Cell cycle (Georgetown, Tex.) · 2019
In vitro (cells) · 2 results
- Molecular basis for the interaction of [Nle4,D-Phe7]melanocyte stimulating hormone with the human melanocortin-1 receptor.
Yang Yk · The Journal of biological chemistry · 1997
In vitro (cells) · 3 results
- Characterization of murine melanocortin receptors mediating adipocyte lipolysis and examination of signalling pathways involved.
Møller CL · Molecular and cellular endocrinology · 2011
In vitro (cells) · mouse · 2 results
- Melanocortin receptor signaling in RAW264.7 macrophage cell line.
Lam CW · Peptides · 2006
In vitro (cells) · mouse · 7 results
- Binding and cAMP studies of melanotropin peptides with the cloned human peripheral melanocortin receptor, hMC1R.
Haskell-Luevano C · Biochemical and biophysical research communications · 1994
In vitro (cells) · 2 results
- Pharmacological comparison of rat and human melanocortin 3 and 4 receptors in vitro.
Schiöth HB · Regulatory peptides · 2002
In vitro (cells) · rat · 1 result
- Temporal cAMP Signaling Selectivity by Natural and Synthetic MC4R Agonists.
Molden BM · Molecular endocrinology (Baltimore, Md.) · 2015
In vitro (cells) · 5 results
- Peptide and small molecules rescue the functional activity and agonist potency of dysfunctional human melanocortin-4 receptor polymorphisms.
Xiang Z · Biochemistry · 2007
In vitro (cells) · 1 result
- Identification of differential melanocortin 4 receptor agonist profiles at natively expressed receptors in rat cortical astrocytes and recombinantly expressed receptors in human embryonic kidney cells.
Selkirk JV · Neuropharmacology · 2007
In vitro (cells) · rat · 2 results
- Melanocortin 4 receptor activation inhibits presynaptic N-type calcium channels in amygdaloid complex neurons.
Agosti F · The European journal of neuroscience · 2014
In vitro (cells) · mouse · 4 results
- Stimulation of intracellular free calcium in GH3 cells by gamma3-melanocyte-stimulating hormone. Involvement of a novel melanocortin receptor?
Langouche L · Endocrinology · 2001
In vitro (cells) · 2 results
- Overexpression and functional characterisation of the human melanocortin 4 receptor in Sf9 cells.
Dolby V · Protein expression and purification · 2004
In vitro (cells) · 1 result
- Rattus norvegicus melanocortin 3 receptor: a corrected sequence.
Daniels D · Peptides · 2005
In vitro (cells) · rattus norvegicus · 1 result
- Effects of pH, salt and time on ligand binding properties of overexpressed melanocortin 4 receptor.
Dolby V · Journal of biochemical and biophysical methods · 2004
In vitro (cells) · 2 results
- Neuropeptide Y-mediated inhibition of proopiomelanocortin neurons in the arcuate nucleus shows enhanced desensitization in ob/ob mice.
Roseberry AG · Neuron · 2004
Other design · mouse · 1 result
- The PVH as a site of CB1-mediated stimulation of thermogenesis by MC4R agonism in male rats.
Monge-Roffarello B · Endocrinology · 2014
Not a test of Melanotan II alone · 14 results
- Type I beta-turn conformation is important for biological activity of the melanocyte-stimulating hormone analogues.
Li SZ · European journal of biochemistry · 1999
Not a test of Melanotan II alone · 9 results
- Biological and conformational study of beta-substituted prolines in MT-II template: steric effects leading to human MC5 receptor selectivity.
Cai M · The journal of peptide research : official journal of the American Peptide Society · 2004
Not a test of Melanotan II alone · 6 results
- Loss of melanocortin receptor accessory protein 2 in melanocortin-4 receptor neurons protect from obesity-associated autonomic and cardiovascular dysfunctions.
Guo DF · Cardiovascular research · 2025
Not a test of Melanotan II alone · 6 results
- Structure-function studies on the cyclic peptide MT-II, lactam derivative of alpha-melanotropin.
Bednarek MA · Peptides · 1999
Not a test of Melanotan II alone · 5 results
- Analogs of MTII, lactam derivatives of alpha-melanotropin, modified at the N-terminus, and their selectivity at human melanocortin receptors 3, 4, and 5.
Bednarek MA · Biochemical and biophysical research communications · 1999
Not a test of Melanotan II alone · 5 results
- Melanoma targeting with alpha-melanocyte stimulating hormone analogs labeled with fac-[99mTc(CO)3]+: effect of cyclization on tumor-seeking properties.
Raposinho PD · Journal of biological inorganic chemistry : JBIC : a publication of the Society of Biological Inorganic Chemistry · 2008
Not a test of Melanotan II alone · 4 results
- A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptides.
Sun H · Bioorganic & medicinal chemistry · 2004
Not a test of Melanotan II alone · 4 results
- Glucose-regulated protein 78 binds to and regulates the melanocortin-4 receptor.
Yoon YR · Experimental & molecular medicine · 2018
Not a test of Melanotan II alone · 4 results
- The stimulatory G protein Gsα is required in melanocortin 4 receptor-expressing cells for normal energy balance, thermogenesis, and glucose metabolism.
Podyma B · The Journal of biological chemistry · 2018
Not a test of Melanotan II alone · 3 results
- NMDA-type glutamate receptors participate in reduction of food intake following hindbrain melanocortin receptor activation.
Campos CA · American journal of physiology. Regulatory, integrative and comparative physiology · 2015
Not a test of Melanotan II alone · 3 results
- Development of Ligand-Drug Conjugates Targeting Melanoma through the Overexpressed Melanocortin 1 Receptor.
Zhou Y · ACS pharmacology & translational science · 2020
Not a test of Melanotan II alone · 3 results
- High-performance liquid chromatographic assay for the alpha-melanotropin[4,10] fragment analogue (Melanotan-II) in rat plasma.
Ugwu SO · Journal of chromatography · 1992
Not a test of Melanotan II alone · 3 results
- Determination of melanotan II in rabbit urine using solid-phase extraction sample preparation followed by reversed-phase high-performance liquid chromatography.
Walters AE · Journal of chromatography. B, Biomedical sciences and applications · 1997
Not a test of Melanotan II alone · 3 results
- Long-term orexigenic effects of AgRP-(83---132) involve mechanisms other than melanocortin receptor blockade.
Hagan MM · American journal of physiology. Regulatory, integrative and comparative physiology · 2000
Not a test of Melanotan II alone · 2 results
- AVP neurons in the paraventricular nucleus of the hypothalamus regulate feeding.
Pei H · Molecular metabolism · 2014
Not a test of Melanotan II alone · 2 results
- A brain leptin-renin angiotensin system interaction in the regulation of sympathetic nerve activity.
Hilzendeger AM · American journal of physiology. Heart and circulatory physiology · 2012
Not a test of Melanotan II alone · 2 results
- Multiple N-methylation of MT-II backbone amide bonds leads to melanocortin receptor subtype hMC1R selectivity: pharmacological and conformational studies.
Doedens L · Journal of the American Chemical Society · 2010
Not a test of Melanotan II alone · 2 results
- Involvement of hypothalamic AMP-activated protein kinase in leptin-induced sympathetic nerve activation.
Tanida M · PloS one · 2013
Not a test of Melanotan II alone · 2 results
- Maternal obesity increases hypothalamic leptin receptor expression and sensitivity in juvenile obesity-prone rats.
Gorski JN · American journal of physiology. Regulatory, integrative and comparative physiology · 2007
Not a test of Melanotan II alone · 2 results
- Three-dimensional molecular models of the hMC1R melanocortin receptor: complexes with melanotropin peptide agonists.
Haskell-Luevano C · Drug design and discovery · 1996
Not a test of Melanotan II alone · 2 results
- Solution structures of cyclic melanocortin agonists and antagonists by NMR.
Ying J · Biopolymers · 2003
Not a test of Melanotan II alone · 2 results
- Analogs of lactam derivatives of alpha-melanotropin with basic and acidic residues.
Bednarek MA · Biochemical and biophysical research communications · 2000
Not a test of Melanotan II alone · 2 results
- Identification and characterization by LC-UV-MS/MS of melanotan II skin-tanning products sold illegally on the Internet.
Breindahl T · Drug testing and analysis · 2015
Not a test of Melanotan II alone · 2 results
- 1H-NMR studies on a potent and selective antagonist at human melanocortin receptor 4 (hMC-4R).
Victoria Silva Elipe M · Biopolymers · 2003
Not a test of Melanotan II alone · 2 results
- Changes of melanocytic lesions inducedby Melanotan injections and sun bed use ina teenage patient with FAMMM syndrome.
Sivyer GW · Dermatology practical & conceptual · 2012
Not a test of Melanotan II alone · 2 results
- Prevalence of mutations and functional analyses of melanocortin 4 receptor variants identified among 750 men with juvenile-onset obesity.
Larsen LH · The Journal of clinical endocrinology and metabolism · 2005
Not a test of Melanotan II alone · 1 result
- Brainstem mechanisms integrating gut-derived satiety signals and descending forebrain information in the control of meal size.
Berthoud HR · Physiology & behavior · 2006
Not a test of Melanotan II alone · 1 result